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2. Muscimol - Wikipedia

   en.wikipedia.org/wiki/Muscimol

   Muscimol is a potent GABA A agonist, activating the receptor for the brain's principal inhibitory neurotransmitter, GABA. Muscimol binds to the same site on the GABA A receptor complex as GABA itself, as opposed to other GABAergic drugs such as barbiturates and benzodiazepines which bind to separate regulatory sites. [ 10 ]

3. Homotaurine - Wikipedia

   en.wikipedia.org/wiki/Homotaurine

   Homotaurine has been reported as a GABA antagonist, [4] as well as a GABA agonist. [10] [11] In vitro studies have found that homotaurine is a GABA A partial agonist [12] as well as a GABA B receptor partial agonist with low efficacy, becoming an antagonist and displacing the full agonists GABA and baclofen at this receptor. [13]

4. Picamilon - Wikipedia

   en.wikipedia.org/wiki/Picamilon

   Picamilon (also known as N-nicotinoyl-GABA, pycamilon, and pikamilon) is a drug formed by a synthetic combination of niacin and γ-aminobutyric acid (GABA). It was developed in the Soviet Union in 1969 [3] and further studied in both Russia [4] and Japan as a prodrug of GABA. [5] In Russia, picamilon is sold as a prescription drug.

5. Phenibut - Wikipedia

   en.wikipedia.org/wiki/Phenibut

   Phenibut is used in Russia, Ukraine, Belarus and Latvia as a pharmaceutical drug to treat anxiety and to improve sleep (e.g., in the treatment of insomnia). [5] [6] It is also used for various other indications, including the treatment of asthenia, depression, alcoholism, alcohol withdrawal syndrome, post-traumatic stress disorder, stuttering, tics, vestibular disorders, Ménière's disease ...

6. Valerenic acid - Wikipedia

   en.wikipedia.org/wiki/Valerenic_acid

   A small study with six human subjects found that valerenic acid peaked in concentration after about an hour and had an average half-life of 1.1 +/- 0.6 hours after oral ingestion of a commercially available valerian root supplement. [8] A later study from the same lab done with sixteen older women found similar values. [3]

7. Gaboxadol - Wikipedia

   en.wikipedia.org/wiki/Gaboxadol

   Gaboxadol is a supra-maximal agonist at α 4 β 3 δ, low-potency agonist at α 1 β 3 γ 2, partial agonist at α 4 β 3 γ, and antagonist at ρ1 GABA A receptors. [5] [6] [7] Its affinity for extrasynaptic α 4 β 3 δ GABA A receptors is 10-fold greater than other subtypes. [8]