enow.com Web Search

  1. Ads

    related to: list of steroid inhibitors for prostate cancer

Search results

  1. Results from the WOW.Com Content Network
  2. Steroidal antiandrogen - Wikipedia

    en.wikipedia.org/wiki/Steroidal_antiandrogen

    Galeterone (TOK-001, VN/124-1): A dual AR antagonist and steroidogenesis inhibitor which was under development for the treatment of prostate cancer but showed insufficient effectiveness in clinical trials and was discontinued. Inocoterone acetate (RU-38882, RU-882): A steroid-like NSAA. It was under development as a topical medication for the ...

  3. Steroidogenesis inhibitor - Wikipedia

    en.wikipedia.org/wiki/Steroidogenesis_inhibitor

    Aromatase inhibitors (AIs) such as aminoglutethimide, anastrozole, exemestane, letrozole, and testolactone inhibit the production of estrogens from androgens and are used mainly in the treatment of estrogen receptor-positive breast cancer. [30] Steroid sulfotransferase (SST) inhibitors prevent the conversion of steroid hormones such as estrone ...

  4. CYP17A1 inhibitor - Wikipedia

    en.wikipedia.org/wiki/CYP17A1_inhibitor

    CYP17A1 inhibitors may inhibit one or both of the enzyme’s functions: 17α-hydroxylase and 17,20-lyase. Some inhibitors are selective and target only the 17,20-lyase function, while others inhibit both functions. [2] By inhibiting these enzymatic functions, CYP17A1 inhibitors prevent the conversion of pregnane steroids into androgens like ...

  5. Antiandrogen - Wikipedia

    en.wikipedia.org/wiki/Antiandrogen

    In addition to active treatment of prostate cancer, antiandrogens are effective as prophylaxis (preventatives) in reducing the risk of ever developing prostate cancer. [32] Antiandrogens have only limitedly been assessed for this purpose, but the 5α-reductase inhibitors finasteride and dutasteride and the steroidal AR antagonist spironolactone ...

  6. List of antiandrogens - Wikipedia

    en.wikipedia.org/wiki/List_of_antiandrogens

    This is a list of antiandrogens, [1] or drugs that prevent the effects of androgens like testosterone and dihydrotestosterone (DHT). [2] It includes direct antagonists of the androgen receptor (AR), androgen synthesis inhibitors like 5α-reductase inhibitors and CYP17A1 inhibitors , and antigonadotropins like GnRH analogues , estrogens , and ...

  7. 5α-Reductase inhibitor - Wikipedia

    en.wikipedia.org/wiki/5α-reductase_inhibitor

    [9] [10] It can also reduce DHT levels in the prostate by 97 to 99% in men with prostate cancer. [11] [12] Epristeride (brand names Aipuliete, Chuanliu) is marketed in China for the treatment of benign prostatic hyperplasia. [13] [14] [15] However, it can only decrease circulating DHT levels by about 25 to 54%. [16]

  1. Ads

    related to: list of steroid inhibitors for prostate cancer