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Typical Oral Dosage Formulations (mg) Approx. Equivalent Oral Dose to 10 mg Diazepam [b] (mg) Peak Onset of Action (hours) Elimination Half-life of Active Metabolite (hours) Primary Therapeutic Use Adinazolam: Deracyn: Research chemical: 1–2: 3: anxiolytic, antidepressant: Alprazolam
[4] [5] Bromazolam is a non subtype selective agonist at the benzodiazepine site of GABA A receptors, with a binding affinity of 2.81 nM at the α 1 subtype, 0.69 nM at α 2 and 0.62 nM at α 5. [6] The "common" dosage range for users of bromazolam was reported to be 1–2 mg, suggesting its potency is similar to alprazolam. [7]
Rilmazafone [1] (リスミー, Rhythmy, previously known as 450191-S) is a water-soluble prodrug developed in Japan. [2] Inside the human body, rilmazafone is converted into several benzodiazepine metabolites that have sedative and hypnotic effects.
Common effects, which vary depending on the substance and dosage in question, may include enhanced alertness, awareness, wakefulness, endurance, productivity, and motivation, increased arousal, locomotion, heart rate, and blood pressure, and the perception of a diminished requirement for food and sleep.
Flubromazolam (JYI-73) [2] [3] [4] is a triazolobenzodiazepine (TBZD), which are benzodiazepine (BZD) derivatives. [5] [6] [7] [8] [9] [10] [11] Flubromazolam is ...
(in doses higher than 10 mg) 7-Nitro-5-phenyl-1,3-dihydro-2H-1,4-benzodiazepin-2-on Nordazepam (in doses higher than 15 mg) 7-Chlor-5-phenyl-1,3-dihydro-2H-1,4-benzodiazepin-2-on Normethadone: 6-Dimethylamino-4,4-diphenyl-hexan-3-on Opium: Oxazepam (in doses higher than 50 mg) 7-Chlor-3-hydroxy-5-phenyl-1,3-dihydro-2H-1,4-benzo-diazepin-2-on ...
Flubrotizolam (2-bromo-4-(2-fluorophenyl)-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine) is a thienotriazolodiazepine derivative with potent sedative and anxiolytic effects, which has been sold as a designer drug.
Felbamate is available in tablets (400 mg and 600 mg) and as a peach-coloured oral suspension (600 mg/5 mL). Adults (≥ 14 years): begin with 1,200 mg daily given every 6 to 8 hours Children (2–14 years): 15 to 45 mg per kg per day given every 6 to 8 hours